Efficacious and rapid metal- and solvent-free synthesis of enantiopure oxazolines

DOI: 10.1016/j.tetasy.2014.08.010

Source and publish data:

Tetrahedron Asymmetry p. 1275 - 1279 (2014)

Update date:2022-08-03

Topics: Isolation and Purification Starting Materials Activation of Carboxylic Acid

Authors:

Hassani, Rym

Requet, Alexandre

Marque, Sylvain

Gaucher, Anne

Prim, Damien

Kacem, Yakdhane

Hassine, Bchir Ben

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Article abstract of DOI:10.1016/j.tetasy.2014.08.010

A rapid and efficient synthesis of oxazolines was performed starting from various nitriles using microwave irradiation combined to metal- and solvent-free conditions to afford high to quantitative yields of the targeted heterocycles.

Full text of DOI:10.1016/j.tetasy.2014.08.010

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