2,3-Dihydro-dithiin and -dithiepine-1,1,4,4-tetroxides: Small molecule non-peptide antagonists of the human galanin hGAL-1 receptor

DOI: 10.1016/S0968-0896(00)00062-6

Source and publish data:

Bioorganic and Medicinal Chemistry p. 1383 - 1391 (2000)

Update date:2022-08-03

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Authors:

Scott, Malcolm K.

Ross, Tina M.

Lee, Daniel H. S.

Wang, Hoau-Yan

Shank, Richard P.

Wild, Kenneth D.

Davis, Coralie B.

Crooke, Jeffrey J.

Potocki, Alexander C.

Reitz, Allen B.

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Article abstract of DOI:10.1016/S0968-0896(00)00062-6

The neuropeptide galanin modulates several physiological functions such as cognition, learning, feeding behavior, and depression, probably via the galanin 1 receptor (GAL-R1). Using an HTS assay based on ¹²⁵I-human galanin binding to the human

Full text of DOI:10.1016/S0968-0896(00)00062-6

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