Bioorganic and Medicinal Chemistry Letters p. 3441 - 3444 (2004)
Update date:2022-08-05
Topics:
Mitchinson, Andrew
Atack, John R.
Blurton, Peter
Carling, Robert W.
Castro, Jose L.
Curley, Karen S.
Russell, Michael G. N.
Marshall, George
McKernan, Ruth M.
Moore, Kevin W.
Narquizian, Robert
Smith, Alison
Street, Leslie J.
Thompson, Sally-Anne
Wafford, Keith
2,5-Dihydropyrazolo[4,3-c]pyridin-3-ones are GABAA receptor benzodiazepine binding site ligands with functional selectivity for the α3 subtype over the α1 subtype. SAR studies to optimise this functional selectivity are described.
View Morewebsite:http://www.tbbmed.com
Contact:86--21-50498136
Address:Room 6002, Building 7-1, No.160 Basheng Road,Pudong Area,Shanghai China
Zhejiang Newfine Industry Co.,Ltd.
Contact:+86-573-82262042
Address:No.225,Dongqing Road, garoms@163.com
Jiaxing Trustworthy Import And Export Co.,Ltd
Contact:+86-573-82030555
Address:Room 1202, Unit B, Charming plaza,No.1558 East Zhongshan Road , Jiaxing City, Zhejiang Province, China.
ShiJiaZhuang Dowell Chemical Co.,Ltd.
website:http://www.dowechem.com
Contact:+86-13463963265
Address:Xiyangling village, high tech Zone, Shijiazhuang,Hebei, China
ShiJiaZhuang Dowell Chemical Co.,Ltd.
website:http://www.dowechem.com
Contact:+86-13463963265
Address:Xiyangling village, high tech Zone, Shijiazhuang,Hebei, China
Doi:10.1016/j.molcata.2015.11.011
(2016)Doi:10.1021/jm960177x
(1996)Doi:10.1063/1.466052
(1993)Doi:10.1002/chem.200700202
(2007)Doi:10.1246/bcsj.50.1980
(1977)Doi:10.1016/j.bmcl.2011.06.041
(2011)