AMIDINOETHYLATION - A NEW REACTION - III; THE AMIDINOETHYLATION OF AMINO-COMPOUNDS: A FACILE SYNTHESIS OF 3-AMINOSUBSTITUTED-N,N'-SUBSTITUTED-PROPANAMIDINES

Article abstract of DOI:10.1016/S0040-4020(01)92361-0

The amidinoethylation of amino compounds takes place by the addition of amines to the C=C double bond of a variety of N,N'-substituted-propenamidines 1.The most nucleophilic amines such as piperidine, morpholine and pyrrolidine add under very smooth condi