Journal of Medicinal Chemistry p. 1137 - 1141 (1984)
Update date:2022-08-02
Topics:
Ogata, Masaru
Matsumoto, Hiroshi
Kida, Shiro
Shiomi, Teruo
Eigyo, Masami
Hirose, Katsumi
A series of some novel N-<(1-ethyl-2-pyrrolidinyl)methyl>benzamides involving replacement of the sulfamoyl group in sulpiride with a sulfonamido group was synthesized and tested for dopamine receptor blockade.In comparison with sulpiride, several compounds were considerably more potent than sulpiride as dopamine receptor blockers.The structure-activity relationships are discussed.
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