Journal of Medicinal Chemistry p. 1137 - 1141 (1984)
Update date:2022-08-02
Topics:
Ogata, Masaru
Matsumoto, Hiroshi
Kida, Shiro
Shiomi, Teruo
Eigyo, Masami
Hirose, Katsumi
A series of some novel N-<(1-ethyl-2-pyrrolidinyl)methyl>benzamides involving replacement of the sulfamoyl group in sulpiride with a sulfonamido group was synthesized and tested for dopamine receptor blockade.In comparison with sulpiride, several compounds were considerably more potent than sulpiride as dopamine receptor blockers.The structure-activity relationships are discussed.
View MoreSuZhou Ascepion Pharmaceuticals, Inc.(expird)
Contact:0512-86881668
Address:Building C,68Xingqing Road,Suzhou,China.
PINGYUAN SIHUAN PHARMACEUTICAL CO., LTD
Contact:+86-531-55696072
Address:#2766,yinxiu Road, Economic Development Zone, Pingyuan Country, Shandong Province, China.
Nanjing Chemzam Pharmtech Co., Ltd.
Contact:+86-25-86462165,+86-13915979898
Address:C5-1，6 Maiyue Road，Maigaoqiao，Nanjing，Jiangsu，China
Contact:86 311 85902108 / 85902109
Address:room 1001-1005 ,huanghe Road ,shijiazhuang ,China
Wuhan Chemwish Technology Co., Ltd
website:http://www.chemwish.com/
Contact:+86-27-67849912
Address:Room 1311, Unit 2, Block1, Innovation Road East Lake High-tech Development Zone Wuhan, Hubei，P.R. China
Doi:10.1021/jo00347a014
(1982)Doi:10.1021/ol0481131
(2004)Doi:10.1023/B:RUBI.0000030129.13466.18
(2004)Doi:10.1002/hc.20111
(2005)Doi:10.1021/ja01122a023
(1952)Doi:10.1055/s-2004-831213
(2004)
