Journal of Medicinal Chemistry p. 1137 - 1141 (1984)
Update date:2022-08-02
Topics:
Ogata, Masaru
Matsumoto, Hiroshi
Kida, Shiro
Shiomi, Teruo
Eigyo, Masami
Hirose, Katsumi
A series of some novel N-<(1-ethyl-2-pyrrolidinyl)methyl>benzamides involving replacement of the sulfamoyl group in sulpiride with a sulfonamido group was synthesized and tested for dopamine receptor blockade.In comparison with sulpiride, several compounds were considerably more potent than sulpiride as dopamine receptor blockers.The structure-activity relationships are discussed.
View MoreJIANGXI ZHANGFENG CHEMICAL CO., LTD.
Contact:+86-0799-3413066
Address:Xiyuan village, Xiabu Town, Xiangdong District
Wuhan Soleado Technology Co.,Ltd.
Contact:86-2783341481 18971291927
Address:RM2405 Unit 1 Builing 1, Taiyin Tower, Changqing Road,Wuhan China
Synochem Ingredients Corp., Ltd.
Contact:+86-512-5636 2180
Address:Zhangjiagang Free Trade Zone
Contact:+86-10-83993285
Address:Rm.1708, Haobai Tower, Building 6, No.50, North Road, West Third Ring, Haidian District, Beijing, China
Xinjiang Zhongtai Chemical Co., Ltd.
Contact:+86-991-8788172
Address:NO.78 XISHAN RD.URUMQI，CHINA
Doi:10.1021/jo00347a014
(1982)Doi:10.1021/ol0481131
(2004)Doi:10.1023/B:RUBI.0000030129.13466.18
(2004)Doi:10.1002/hc.20111
(2005)Doi:10.1021/ja01122a023
(1952)Doi:10.1055/s-2004-831213
(2004)
