Three-component synthesis of polysubstituted 6-azaindolines and its tricyclic derivatives

DOI: 10.1021/ol0477881

Source and publish data:

Organic Letters p. 239 - 242 (2005)

Update date:2022-08-04

Topics:

Authors:

Fayol, Aude

Zhu, Jieping

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Article abstract of DOI:10.1021/ol0477881

(Chemical Equation Presented) By simply heating a toluene solution of isocyanoacetamide (3), amine (4), and aldehyde (5), a clean three-component reaction occurred to provide the pyrrolidinone-fused azaindoline (2). In this multicomponent reaction, the is

Full text of DOI:10.1021/ol0477881

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