Application of intramolecular 1,3-dipolar cyclic addition of azide and olefin; Construction of (pyrrolidine-2-ylidene)glycinate and glycinamides

DOI: 10.1248/cpb.53.529

Source and publish data:

Chemical and Pharmaceutical Bulletin p. 529 - 536 (2005)

Update date:2022-08-03

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Authors:

Konda-Yamada, Yaeko

Asano, Keiko

Satou, Takahiro

Monma, Souichi

Sakayanagi, Masataka

Satou, Noriko

Takeda, Kazuyoshi

Harigaya, Yoshihiro

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Article abstract of DOI:10.1248/cpb.53.529

Oxopropyl E-(pyrrolidine-2-ylidene)glycinamide (5c) and allyl E-(pyrrolidine-2-ylidene)glycinate (5d) were effectively synthesized from 2,3,5-tri-O-benzyl-4-O-tert-butyldimethylsilyl(TBDMS)-D-arabinal (7) using intramolecular 1,3-dipolar cyclic reaction o

Full text of DOI:10.1248/cpb.53.529

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Product name:methyl (E,3R,4R,5S)-N-benzyloxycarbonyl-N-tert-butoxycarbonyl-α-(3,4-dibenzyloxy-5-benzyloxymethylpyrrolidin-2-ylidene)glycinate

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