Synthesis and pharmacological characterization of (±)-5,9α-dimethyl-2-[2-(4-fluorophenyl)ethyl]-2'-hydroxy-6,7-benzomor phan (fluorophen), a ligand suitable for visualization of opiate receptors in vivo

DOI: 10.1021/jm00365a017

Source and publish data:

Journal of Medicinal Chemistry p. 1643 - 1645 (1983)

Update date:2022-08-02

Topics:

Authors:

Rice Rice

Konicki Konicki

Quirion Quirion

Burke Jr.

Pert Pert

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1021/jm00365a017

A fluorinated derivative of the benzomorphan opiate agonist phenazocine, (±)-5,9α-dimethyl-2-[2-(4-fluorophenyl)ethyl-2'-hydroxy-6,7-benzomorphan (fluorophen), was prepared by N-acylation of (±)-5,9α-dimethyl-2'-hydroxybenzomorphan with (p-fluorophenyl)ac

Full text of DOI:10.1021/jm00365a017

Products guided by the article

Product name:2-(4-Fluoro-phenyl)-1-((2R,6R,11R)-8-hydroxy-6,11-dimethyl-1,2,5,6-tetrahydro-4H-2,6-methano-benzo[d]azocin-3-yl)-ethanone

Cas No:86436-93-3

R&D Labs maybe for 86436-93-3

Shanghai Forever Synthesis Co.,Ltd.

Contact:021-61124658

Address:Zhoukang Road,Pudong New District,Shanghai,China
Shandong Shouguang Songchuan Industrial Additives Co.,Ltd

Contact:+86-536-8566856

Address:Shouguang,Shandong,China
Zhejiang kehong chemical co., ltd

Contact:0086-575-85522000

Address:xiner center RD binhai industrial zone shaoxing zhejiang province P.R.China,312073
Qingdao Pana-Life Biochem Co.,Ltd.

Contact:86-532-87683902

Address:No.967 Dalao Road, Licang Zone, Qingdao City,Shandong, China 266021
Anhui Biochem United Pharmaceutical Co., Ltd.

Contact:0086 551 5167062 / 5228268

Address:No. 30 Hongfeng Road, Hi-Tech Development Zone, Hefei (230088), China

Relevant to this article

Chiral recognition by CD-sensitive dimeric zinc porphyrin host. 1. Chiroptical protocol for absolute configurational assignments of monoalcohols and primary monoamines

Doi:10.1021/ja010249w
(2001)
Stibasilene Sb-Si and its lighter homologues: A comparative study

Doi:10.1021/ja5026084
(2014)
A PRACTICAL AND CONVENIENT SYNTHESIS OF THE NITROETHYLENE TRANSFER REAGENT, 2-NITROETHYL PHENYL SULFOXIDE

Doi:10.1016/S0040-4039(00)96237-3
(1987)
A convenient and new approach to the synthesis of ω-heterocyclic amino acids from carboxy lactams through ring-chain-transformation. Part 2: Synthesis of (2R)-/(2S)-2-aminomethyl-3-(1-aryl-/1,5-diaryl-1H-pyrazol-3-yl)- propionic acid

Doi:10.1016/j.tet.2005.07.018
(2005)
Photophysical properties of borondipyrromethene analogues in solution

Doi:10.1021/jp052626n
(2005)
AMIDOALKYLATION OF DIENES WITH ADDUCTS OF GLYOXYLIC ACID - SYNTHESIS OF α-ACYLAMINO-γ-ALKENYL-γ-BUTYROLACTONES

Doi:10.1016/S0040-4039(00)81575-0
(1983)

Article Doi