Bioorganic and Medicinal Chemistry Letters p. 386 - 390 (2008)
Update date:2022-08-05
Topics:
Dai, Yujia
Hartandi, Kresna
Soni, Niru B.
Pease, Lori J.
Reuter, David R.
Olson, Amanda M.
Osterling, Donald J.
Doktor, Stella Z.
Albert, Daniel H.
Bouska, Jennifer J.
Glaser, Keith B.
Marcotte, Patrick A.
Stewart, Kent D.
Davidsen, Steven K.
Michaelides, Michael R.
Tumor angiogenesis is mediated by KDR and other VEGFR and PDGFR kinases. Their inhibition presents an attractive approach for developing anticancer therapeutics. Here, we report a series of aminopyrazolopyridine ureas as potent VEGFR/PDGFR multitargeted k
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