Bioorganic and Medicinal Chemistry Letters p. 5474 - 5477 (2005)
Update date:2022-08-03
Topics:
Pan, Weitao
Liu, Hu
Xu, Yong-Jiang
Chen, Xin
Kim, Ki Hwan
Milligan, Daniel L.
Columbus, John
Hadari, Yaron R.
Kussie, Paul
Wong, Wai C.
Labelle, Marc
Pyrimido-oxazepine based sub-micromolar inhibitors (2-4) for Aurora and FLT-3 were designed and synthesized. These preliminary results supported the potential use of pyrimido-oxazepines as a versatile template for developing specific kinase inhibitors.
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