Conformationally Restrained Fentanyl Analogues. 2. Synthesis and Analgetic Evaluation of Perhydro-1,6-naphthyridin-2-ones

DOI: 10.1021/jm00376a007

Source and publish data:

Journal of Medicinal Chemistry p. 1271 - 1275 (1984)

Update date:2022-08-04

Topics:

Authors:

Borne, Ronald F.

Fifer, E. Kim

Waters, I.W.

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1021/jm00376a007

Conformational flexibility of the N-acyl portion of fentanyl-type analgetics was restricted through the synthesis of novel perhydro-1,6-naphthyridin-2-one derivatives.Neither the cis-fused derivative (5a), the trans-fused derivative (5b), nor the enamide

Full text of DOI:10.1021/jm00376a007

Products guided by the article

Product name:Pyridine, 1,2,3,6-tetrahydro-1-(2-phenylethyl)-4-(1-pyrrolidinyl)-

Cas No:91157-36-7

R&D Labs maybe for 91157-36-7

Jinzhou Jiutai Pharmaceutical Co.,Ltd

Contact:+86-0416-5179890

Address:No.41, Taianli, Taihe District, Jinzhou, Liaoning
sichuan tiancai fine co LTD.

website:http://www.tcfinechem.com/

Contact:18681346930

Address:baifu town,whou district
Zhejiang Chemicals Import & Export Corporation

Contact:86-571-87043088

Address:No.37,Qingchun Road,Hangzhou,China
Deer Chemicals Co., Ltd.

Contact:+86-13666670345

Address:Agricultural Development Zone, Haining, Jiaxing, Zhejiang
FREEBARQUE DEVELOPMENT GROUP LIMITED

Contact:+86(0)10-5109 5335 or 5109 5345

Address:Room602,Block1-B,LINGDI OFFICE,NO.13 BEIYUAN ROAD

Relevant to this article

SYNTHESES AND SPECTROSCOPIC STUDIES ON SOME PLATINUM GROUP METAL COMPLEXES WITH OXAZEPAM AS LIGAND

Doi:10.1016/0022-2860(84)87050-7
(1984)
The One-Electron Transfer Induced Photocycloreversion of Stilbazolium Cyclodimers

Doi:10.1246/bcsj.71.419
(1998)
Total Synthesis of a Partial Structure from Arabinogalactan and Its Application for Allergy Prevention

Doi:10.1002/chem.202002287
(2021)
Trigonal-bipyramidal geometry induced by an external water ligand in a sterically hindered iron salen complex, related to the active site of protocatechuate 3,4-dioxygenase

Doi:10.1021/ic060650p
(2006)
Synthesis of Lewis A trisaccharide analogues in which d-glucose and l-rhamnose replace d-galactose and l-fucose, respectively

Doi:10.1016/j.carres.2006.07.006
(2006)
Towards a better understanding of photo-excited spin alignment processes using silole diradicals

Doi:10.1039/b606593g
(2006)

Article Doi