Identification of a novel boron-containing antibacterial agent (AN0128) with anti-inflammatory activity, for the potential treatment of cutaneous diseases

DOI: 10.1016/j.bmcl.2006.08.130

Source and publish data:

Bioorganic and Medicinal Chemistry Letters p. 5963 - 5967 (2006)

Update date:2022-08-02

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Authors:

Baker, Stephen J.

Akama, Tsutomu

Zhang, Yong-Kang

Sauro, Vittorio

Pandit, Chetan

Singh, Rajeshwar

Kully, Maureen

Khan, Jehangir

Plattner, Jacob J.

Benkovic, Stephen J.

Lee, Ving

Maples, Kirk R.

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Article abstract of DOI:10.1016/j.bmcl.2006.08.130

A series of borinic acid picolinate esters were synthesized and screened for their minimum inhibitory concentration (MIC) against Gram-positive and -negative bacteria. Our lead compounds were then screened for anti-inflammatory activity. From these studie

Full text of DOI:10.1016/j.bmcl.2006.08.130

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