Tetrahedron Letters p. 841 - 844 (1980)
Update date:2022-09-26
Topics:
Nagao, Yoshimitsu
Seno, Kaoru
Kawabata, Kohji
Miyasaka, Tadayo
Takao, Sachiko
Fujita, Eiichi
3-Acylthiazolidine-2-thiones (1) were easily prepared and they were treated with several amines in dichloromethane to give amides 4 in very high yields within a short time.Aminoalcohols and aminophenols were selectively converted into acylaminoalcohols and acylaminophenols, respectively, by this reaction.One can monitor the reaction by disappearance of the yellow color of the starting material 1.Some amide alkaloids (15-18) have effectively been synthesized.
View MoreShangHai Original Economy-Trade Develop Co.,Ltd.,
Contact:86-21-68552131
Address:shanghai
Shanghai Yurui Biotechnology(Anyang) Pharmaceutical Co., Ltd
Contact:+86-0372-3662335 +86-0372-3661988
Address:hanling industrial park anyang
Contact:+86-532-80762375
Address:No. 6, Hongkong Middle Road, Qingdao, China
Qingdao S. H. Huanyu Imp. & Exp. Co., Ltd.
Contact:86-532-88250866
Address:Room 615, World Trade Centre Building B, Hongkong Middle Roda 6#, Qingdao, Shandong, China
Jiangsu Taihu New Materials Holding Co., Ltd
Contact:+86-519-86160108
Address:Xueyan Town, Changzhou City, Jiangsu Province, 213169, China
Doi:10.1016/j.jcat.2017.08.013
(2017)Doi:10.1080/00397911.2017.1382535
(2017)Doi:10.1007/BF00773017
(1984)Doi:10.1021/jo01044a043
(1963)Doi:10.1039/b700852j
(2007)Doi:10.1021/ja01107a046
()