Journal of Medicinal Chemistry p. 1492 - 1500 (2016)
Update date:2022-09-26
Topics:
Baud, Matthias G. J.
Lin-Shiao, Enrique
Zengerle, Michael
Tallant, Cynthia
Ciulli, Alessio
We describe new synthetic routes developed toward a range of substituted analogues of bromo and extra-terminal (BET) bromodomain inhibitors I-BET762/JQ1 based on the triazolo-benzodiazepine scaffold. These new routes allow for the derivatization of the me
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