Selective demethylation and demethoxy-thioalkylation of 5-methoxyindoles

Article abstract of DOI:10.1080/00397919408010187

Under appropriate conditions, hard acid and soft nucleophile system lead to selective demethylation and demethoxy-thioalkylation of certain 5-methoxyindoles.

Full text of DOI:10.1080/00397919408010187

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Synthetic Communications: An
International Journal for Rapid
Communication of Synthetic
Organic Chemistry
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Selective Demethylation and
Demethoxy Thioalkylation of 5-
Methoxyindoles
a
a
Catherine Caubère , Paul Caubère , Pierre Renard
b
b
,
Jean-Guy Bizot-Espiart & Brigitte Jamart-
a
Grègoire
a
Laboratoire de Chimmie Organique I , Unité
Associée au CNRS, Université de Nancy I , BP 239,
F-54506, Vandoeuvre-les-Nancy, France
b
Adir , 1 Rue Carle Hébert, 92415, Courbevoie,
France
Published online: 23 Sep 2006.
To cite this article: Catherine Caubère , Paul Caubère , Pierre Renard , Jean-
Guy Bizot-Espiart & Brigitte Jamart-Grègoire (1994) Selective Demethylation and
Demethoxy Thioalkylation of 5-Methoxyindoles, Synthetic Communications: An
International Journal for Rapid Communication of Synthetic Organic Chemistry, 24:13,
1799-1808, DOI: 10.1080/00397919408010187
To link to this article: http://dx.doi.org/10.1080/00397919408010187
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