Reaction of mercaptoacetate and halides containing activated methylenes with thiocarbamoylimidates: A novel approach to the synthesis of aminothiazole derivatives

Article abstract of DOI:10.1080/00397919808005086

The reaction of N-thiocarbamoylimidates 1 with methyl thioglycolate leads to the formation of 4-arylamino-5-methoxycarbonylthiazoles 2. The condensation of the same imidates 1 on ethyl bromoacetate, benzyl bromide and chloroacetonitrile provides the corre

Full text of DOI:10.1080/00397919808005086

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Synthetic Communications: An
International Journal for Rapid
Communication of Synthetic
Organic Chemistry
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Reaction of Mercaptoacetate
and Halides Containing
Activated Methylenes with
Thiocarbamoylimidates:
A Novel Approach to the
Synthesis of Aminothiazole
Derivatives
a
a
a
K. Dridi , M. L. EL Efrit , B. Baccar & H. Zantour
a
a
Laboratoire de Synthèse Organique, Département
de Chimie, Faculté des Sciences, Campus
Universitaire, 1060, Tunis-Tunisie
Available online: 20 Aug 2006
To cite this article: K. Dridi, M. L. EL Efrit, B. Baccar & H. Zantour (1998):
Reaction of Mercaptoacetate and Halides Containing Activated Methylenes with
Thiocarbamoylimidates: A Novel Approach to the Synthesis of Aminothiazole
Derivatives, Synthetic Communications: An International Journal for Rapid
Communication of Synthetic Organic Chemistry, 28:1, 167-174
To link to this article: http://dx.doi.org/10.1080/00397919808005086
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