REACTION OF IN SITU GENERATED α,β-UNSATURATED IMINES WITH CH-NUCLEOPHILES: A NOVEL AND EFFICIENT SYNTHESIS OF PYRIDINES.

Article abstract of DOI:10.1016/0040-4039(95)02006-B

A novel and highly efficient procedure for the synthesis of 2,4,6-trisubstituted and 2,3,4,6-tetrasubstituted pyridines has been developed.It is based on the one-pot reaction of situ generated α,β-unsaturated imines with CH-nucleophiles.