Tetrahedron Letters p. 9685 - 9688 (1998)
Update date:2022-08-16
Topics:
Chayer, Said
Schmitt, Martine
Collot, Valerie
Bourguignon, Jean-Jacques
Direct acylation of imidazo [1,2-a] pyridines in a sealed tube at 130°C and without catalyst gave various 3-acyl derivatives in satisfactory yields.
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