101248-32-2Relevant academic research and scientific papers
Folate receptor binding conjugates of antifolates
-
Page/Page column 30, (2015/12/04)
Conjugates of antifolates, releasable linkers, and drugs, and pharmaceutical compositions containing them are described. The conjugates are useful for treating diseases arising from pathogenic cell populations. Methods for treating such diseases are also described.
Anti-cancer compounds
-
, (2008/06/13)
Quinazolines of the formula: STR1 wherein R1 -R8 are defined as in the specification, or a pharmaceutically acceptable salt, ester or amide thereof areof therapeutic value, particularly in the treatment of cancer.
Folate Analogues. 26. Syntheses of Antifolate Activity of 10-Substituted Derivatives of 5,8-Dideazafolic Acid and of the Poly-γ-glutamyl Metabolites of N10-Propargyl-5,8-Dideazafolic Acid (PDDF)
Nair, M.G.,Nanavati, Nitin T.,Nair, Indira G.,Kisliuk, Roy L.,Gaumont, Y.,et al.
, p. 1754 - 1760 (2007/10/02)
The poly-γ-glutamyl derivatives of N10-propargyl-5,8-dideazafolic acid (PDDF) with a chain length of up to five glutamate residues were synthesized from N10-propargyl-5,8-dideazapteroic acid (7) by the solid-phase procedure.These com
