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Usage

Uses

Used in Organic Synthesis:
Tert-Butyl 5-methoxy-4-methylpyridin-3-ylcarbamate serves as a reagent in organic synthesis, where its specific structural features contribute to the formation of various complex organic molecules. Its utility in this field is attributed to its ability to participate in a range of chemical reactions, facilitating the synthesis of desired products.
Used in Pharmaceutical Research:
In the pharmaceutical industry, tert-Butyl 5-methoxy-4-methylpyridin-3-ylcarbamate is utilized for research purposes. Its unique structure positions it as a potential candidate for the development of new drugs. tert-Butyl 5-methoxy-4-methylpyridin-3-ylcarbamate's properties may allow it to interact with biological targets in ways that could lead to therapeutic benefits.
Used in Drug Development:
The potential applications of tert-Butyl 5-methoxy-4-methylpyridin-3-ylcarbamate extend to the development of new drugs. Its structural components may offer advantages in medicinal chemistry, such as enhancing the compound's pharmacokinetic or pharmacodynamic profiles, which are critical for drug efficacy and safety.
Used in Agrochemical Development:
Similarly, the compound may also find applications in the agrochemical sector. Its unique structure and properties could be harnessed in the design of new agrochemicals, potentially leading to more effective and targeted pest control solutions.

Upstream product

• 74-88-4 methyl iodide 
• 342603-10-5 tert-butyl 5-methoxypyridin-3-ylcarbamate 
• 64436-92-6 3-amino-5-methoxypyridine 
• 50720-12-2 3-bromo-5-methoxypyridine 

Downstream Products

• 1185094-00-1 3-amino-5-methoxy-4-methylpyridine hydrochloride 
• 1192255-92-7 (3-methoxy[1,5]naphthyridin-4-yl)methanol 
• 1056877-13-4 3-methoxy-1,5-naphthyridine-4-carbaldehyde 
• 1056877-14-5 3-hydroxy[1,5]naphthyridine-4-carbaldehyde 
• 1192256-10-2 3-descladinosyl-11,12-dideoxy-6-O-methyl-3-oxo-12,11-(oxycarbonyl-(1-((3-hydroxy-[1,5]naphthyridin-4-yl)-methyl)-azetidin-3-yl)-imino)-erythromycin A tosylate 

Relevant academic research and scientific papers

Discovery of azetidinyl ketolides for the treatment of susceptible and multidrug resistant community-acquired respiratory tract infections

Respiratory tract bacterial strains are becoming increasingly resistant to currently marketed macrolide antibiotics. The current alternative telithromycin (1) from the newer ketolide class of macrolides addresses resistance but is hampered by serious safe

Process development of a novel azetidinyl ketolide antibiotic

Process development and the multikilogram synthesis of a novel azetidinyl ketolide antibiotic is described. Starting with clarithromycin, the eight-step synthesis features several telescoped operations and direct isolations, which results in a significant improvement in throughput and a major reduction in solvent usage and waste stream volume over the first scale-up campaign. Particular highlights of this effort include the development of an efficient synthesis of 3-hydroxy-1,5-naphthyridine-4-carbaldehyde via a Skraup process and engineering a robust final API synthesis. We also discovered a crystalline monotosylate salt that addressed significant formulation and degradation issues experienced when using the noncrystalline freebase.