1053417-60-9Relevant articles and documents
Novel structure-activity relationships and selectivity profiling of cage dimeric 1,4-dihydropyridines as multidrug resistance (MDR) modulators
Coburger, Claudius,Wollmann, Joerg,Krug, Martin,Baumert, Christiane,Seifert, Marianne,Molnar, Josef,Lage, Hermann,Hilgeroth, Andreas
experimental part, p. 4983 - 4990 (2010/09/10)
Synthesized series of cage dimeric 1,4-dihydropyridines have been systematically evaluated as MDR modulators in in vitro assays to investigate structure-dependent selectivity properties of inhibiting most cancer-relevant efflux pump proteins. Structure-ac