1220529-82-7Relevant academic research and scientific papers
Radiolabeled Dibenzodiazepinone-Type Antagonists Give Evidence of Dualsteric Binding at the M2 Muscarinic Acetylcholine Receptor
Pegoli, Andrea,She, Xueke,Wifling, David,Hübner, Harald,Bernhardt, Günther,Gmeiner, Peter,Keller, Max
, p. 3314 - 3334 (2017/05/05)
The dualsteric ligand approach, aiming at ligands with improved subtype selectivity, has been increasingly applied to muscarinic receptors (MRs). In this article, we present the synthesis and characterization of a M2R subtype-preferring radiola
POTENT AND SELECTIVE INHIBITORS OF NAV1.7
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, (2016/02/18)
Disclosed is a composition of matter comprising an isolated polypeptide, which is a peripherally-restricted NaV1.7 inhibitor. In some disclosed embodiments, the isolated polypeptide is an inhibitor of NaV1.7. Other embodiments are co
Introduction of functionalized mesopores to metal-organic frameworks via metal-ligand-fragment coassembly
Park, Jinhee,Wang, Zhiyong U.,Sun, Lin-Bing,Chen, Ying-Pin,Zhou, Hong-Cai
supporting information, p. 20110 - 20116 (2013/02/23)
Introduction of functionalized mesopores into microporous metal-organic frameworks (MOFs) can endow them with suitable properties for applications in gas storage, separation, catalysis, and drug delivery. However, common methods for functionalization (inc
