1258238-85-5Relevant articles and documents
Preparation of Building Blocks for Iterative Suzuki-Miyaura Reactions via Direct Bromination of Aryl Boronic Acids: One-Pot Total Syntheses of Dictyoterphenyls A and B
Lee, Chun-Young,Cheon, Cheol-Hong
, p. 3831 - 3836 (2017)
A highly efficient method for the preparation of 4-alkoxy-3-bromophenyl boronic acid N-methyliminodiacetic acid (MIDA) esters as building blocks in iterative Suzuki-Miyaura reactions from the 4-alkoxyphenylboronic acids is described using a boronic acid m
Radical C?N Borylation of Aromatic Amines Enabled by a Pyrylium Reagent
Chabbra, Sonia,Cornella, Josep,Leutzsch, Markus,Ma, Yuanhong,Niski, Jan,Pang, Yue,Reijerse, Edward J.,Schnegg, Alexander
supporting information, (2020/03/23)
Herein, we report a radical borylation of aromatic amines through a homolytic C(sp2)?N bond cleavage. This method capitalizes on a simple and mild activation via a pyrylium reagent (ScPyry-OTf) thus priming the amino group for reacti