129398-27-2Relevant academic research and scientific papers
Synthesis of fluorine-containing cyclic α-amino acid and α-amino phosphonate derivatives by alkene metathesis
Osipov, Sergey N.,Artyushin, Oleg I.,Kolomiets, Alexey F.,Bruneau, Christian,Picquet, Michel,Dixneuf, Pierre H.
, p. 3891 - 3897 (2007/10/03)
The electrophilic imino esters XF2CC(=NPG)CO2Me and imino phosphonates CF3CC(=NPG)P(O)(OR)2 (PG = SO2Ph, Cbz, Boc) were transformed by nucleophilic and then electrophilic additions into fluorine-conta
Synthesis, structure and biological activity of α-trifluoromethyl-substituted thyreotropin releasing hormone
Koksch, Beate,Ullmann, Dirk,Jakubke, Hans-Dieter,Burger, Klaus
, p. 53 - 57 (2007/10/03)
The incorporation of α-trifluoromethyl pyroglutamic acid into thyreotropin releasing hormone TRH, results in the complete stability of the pGlu-His bond against proteolytic degradation by pyroglutamyl aminopeptidase II. The influence of the trifluoromethy
