130632-09-6Relevant academic research and scientific papers
Synthesis of novel N-sulfonyl monocyclic β-lactams as potential antibacterial agents
Jarrahpour, Aliasghar,Zarei, Maaroof
, p. 49 - 58 (2006)
New cis monocyclic β-lactams were synthesized by [2+2] Staudinger cycloaddition reactions of the imine (3,4-dimethoxybenzylidene)-(4- methoxyphenyl)amine and ketenes derived from different acyl chlorides and Et3N. These monocyclic β-lactams wer
Catalytic Asymmetric γ-Lactam Synthesis from Enolisable Anhydrides and Imines
Collar, Aarón Gutiérrez,Trujillo, Cristina,Lockett-Walters, Bruce,Twamley, Brendan,Connon, Stephen J.
, p. 7275 - 7279 (2019/05/15)
An anion-binding approach to the problem of preparing enantioenriched γ-lactams from enolisable anhydrides and imines is reported. A simple bisurea catalyst promotes the cycloaddition between α-aryl succinic anhydrides and either PMP- or benzhydryl-protec
Application of a catalyst-free Domino Mannich/Friedel-Crafts alkylation reaction for the synthesis of novel tetrahydroquinolines of potential antitumor activity
Castillo, Juan-Carlos,Jiménez, Elizabeth,Portilla, Jaime,Insuasty, Braulio,Quiroga, Jairo,Moreno-Fuquen, Rodolfo,Kennedy, Alan R.,Abonia, Rodrigo
, p. 932 - 947 (2018/02/09)
A useful and efficient method to construct diversely substituted 1,2,3,4-tetrahydroquinolines in good to excellent yields has been developed through a catalyst-free Domino Mannich and intramolecular Friedel-Crafts alkylation reactions of N-arylamines with
Electroreductive acylation of aromatic imines with acylimidazoles
Kise, Naoki,Morimoto, Shinji
, p. 1765 - 1771 (2008/09/18)
The intermolecular reductive coupling of aromatic imines with acylimidazoles was effected by electroreduction in the presence of chlorotrimethylsilane and gave α-amino-α-aryl ketones. This method was also effective for the synthesis of α-amino-α-aryl esters using methoxycarbonylimidazole as an electrophile.
Transformation of (+)-thiomicamine into a new ligand for the enantioselective addition of methyllithium to prochiral imines
Broezda, Danuta,Chrzanowska, Maria,Glaszynska, Agata,Rozwadowska, Maria D.
, p. 4791 - 4796 (2007/10/03)
A new ligand 2 was prepared from (+)-thiomicamine 1 and o-methoxyphenol, and its activity as an external controller of stereochemistry in enantioselective additions of methyllithium to prochiral imines 8-10 tested. The non-racemic secondary amines 11-13 w
