1312447-85-0Relevant academic research and scientific papers
A one-pot "back-to-front" approach for the synthesis of benzene ring substituted indoles using allylboronic acids
Karan, Ganesh,Sahu, Samrat,Maji, Modhu Sudan
supporting information, p. 5274 - 5277 (2021/06/06)
Synthesis of only benzene ring functionalized indoles and poly-substituted carbazoles is reported via a one-pot triple cascade benzannulation protocol. Usage of differently substituted and readily accessible allylboronic acids as a 3-carbon annulating partner enables diverse aliphatic and aromatic substitution patterns, which is still a daunting task. This scalable synthetic protocol tolerates broad scope, thus enabling further downstream modifications. As an application, carbazole based natural products glycozoline and glycozolinol were synthesized. This journal is
Substituent-Guided Palladium-Ene Reaction for the Synthesis of Carbazoles and Cyclopenta[ b]indoles
Yadav, Sonu,Hazra, Raju,Singh, Animesh,Ramasastry
, (2019/05/07)
An efficient palladium-catalyzed intramolecular Trost-Oppolzer type Alder-ene strategy was developed for the synthesis of carbazoles and cyclopenta[b]indoles from easily accessible(3-allyl-1H-indol-2-yl)methyl acetates. This strategy was extended for the synthesis of naphthalenes and dibenzobenzofurans as well. In addition, a short synthesis of antibacterial and antifungal natural product glycozoline and its analogues was also achieved.
Substituent-Guided Palladium-Ene Reaction for the Synthesis of Carbazoles and Cyclopenta[b]indoles
Yadav, Sonu,Hazra, Raju,Singh, Animesh,Ramasastry
supporting information, p. 2983 - 2987 (2019/05/10)
An efficient palladium-catalyzed intramolecular Trost-Oppolzer type Alder-ene strategy was developed for the synthesis of carbazoles and cyclopenta[b]indoles from easily accessible(3-allyl-1H-indol-2-yl)methyl acetates. This strategy was extended for the synthesis of naphthalenes and dibenzobenzofurans as well. In addition, a short synthesis of antibacterial and antifungal natural product glycozoline and its analogues was also achieved.
Pd-catalyzed intramolecular oxidative C-H amination: Synthesis of carbazoles
Youn, So Won,Bihn, Joon Hyung,Kim, Byung Seok
supporting information; experimental part, p. 3738 - 3741 (2011/09/13)
A Pd-catalyzed oxidative C-H amination of N-Ts-2-arylanilines under ambient temperature using Oxone as an inexpensive, safe, and easy-to-handle oxidant has been developed. This process represents a green and practical method for the facile construction of carbazoles with a broad substrate scope and wide functional group tolerance.
