13207-53-9Relevant articles and documents
Synthesis, characterization and biological activity of some dithiourea derivatives
Frost, Carminita,Hoppe, Heinrich,Hosten, Eric,Isaacs, Michelle,Khanye, Setshaba D.,Krause, Jason,Lobb, Kevin,Odame, Felix,Sayed, Yasien,Tshentu, Zenixole
, p. 764 - 777 (2020/10/02)
Novel dithiourea derivatives have been designed as HIV-1 protease inhibitors using Autodock 4.2, synthesized and characterized by spectroscopic methods and microanalysis. 1-(3-Bromobenzoyl)-3-[2-({[(3-bromophenyl)formami-do]methanethioyl}amino)phenyl]thio
Bioorthogonal Click and Release Reaction of Iminosydnones with Cycloalkynes
Bernard, Sabrina,Audisio, Davide,Riomet, Margaux,Bregant, Sarah,Sallustrau, Antoine,Plougastel, Lucie,Decuypere, Elodie,Gabillet, Sandra,Kumar, Ramar Arun,Elyian, Jijy,Trinh, Minh Nguyet,Koniev, Oleksandr,Wagner, Alain,Kolodych, Sergii,Taran, Frédéric
supporting information, p. 15612 - 15616 (2017/12/02)
We report the discovery of a new bioorthogonal click-and-release reaction involving iminosydnones and strained alkynes. This transformation leads to two products resulting from the ligation and fragmentation of iminosydnones under physiological conditions. Optimized iminosydnones were successfully used to design innovative cleavable linkers for protein modification, thus opening up new areas in the fields of drug release and target-fishing applications. This click-and-release technology offers the possibility of exchanging tags on proteins for functionalized cyclooctynes under mild and bioorthogonal conditions.
ACCELERATORS FOR CURABLE COMPOSITIONS
-
Paragraph 0058, (2014/01/17)
Benzoylthiourea or benzoylthiourethane derivatives as cure accelerators for curable compositions are provided.
ACCELERATORS FOR TWO PART CURABLE COMPOSITIONS
-
Paragraph 0058, (2014/01/17)
Benzoylthiourea or benzoylthiourethane derivatives as cure accelerators for two part curable compositions are provided.
Colorimetric chemosensors designed to provide high sensitivity for Hg 2+ in aqueous solutions
Lin, Qi,Fu, Yong-Peng,Chen, Pei,Wei, Tai-Bao,Zhang, You-Ming
, p. 1 - 6 (2012/11/07)
The specific colorimetric detection of Hg2+ in the context of interference from coexisting metal ions in aqueous solutions is a challenge. Therefore, a series of easy-to-make Hg2+ colorimetric chemosensors S1~S3, bearing thiourea moi
STRUCTURE INVESTIGATIONS ON SOME DIPHENYLTRIAZOLES
Somorai, T.,Dvortsak, P.,Lango, J.,Reiter, J.
, p. 23 - 28 (2007/10/02)
Syntheses of 1,3-diphenyl-4H-1,2,4-triazolin-5-thione (1) and 1,5-diphenyl-2H-1,2,4-triazolin-3-thione (2) have been reinvestigated and the structures proposed in the literature corrected. 1H-NMR, 13C-NMR, UV and MS studies of these compounds and their S-