134357-05-4Relevant academic research and scientific papers
A novel route to N-alkylated derivatives of aziridine-2-carboxylic acid. An alternative synthesis of (S,S)-Bz-Azy-Val-OMe
Polyak,Dorofeeva,Sturkovich,Goldberg
, p. 239 - 248 (1991)
A novel method for N-alkylation of azyridine-2-carboxylic acid derivative with benzyl chloride under phase-transfer conditions or using KF/Al2O3 as a base was developed. The latter variant of this method was applied to carry out the key step of the alternative synthesis of the dipeptide (S,S)-Bz-Azy-Val-Ome.
