1438414-73-3Relevant articles and documents
2,3-Difunctionalized Indoles via Radical Acylation or Trifluoromethylation of ortho-Alkynylphenyl Isonitriles
Leifert, Dirk,Weidlich, Frauke,Adler, Florin,Daniliuc, Constantin G.,Alasmary, Fatmah A.,Studer, Armido
supporting information, p. 284 - 288 (2021/12/27)
A radical cascade to 2,3-disubstituted indoles proceeding via acylation or trifluoromethylation of ortho-alkynylphenyl isonitriles is presented. In these cascades, two C–C bonds and one C–O bond are formed using an inexpensive oxidant and a catalytic copp
Syntheses of N-Alkyl 2-Arylindoles from Saturated Ketones and 2-Arylethynylanilines via Cu-Catalyzed Sequential Dehydrogenation/Aza-Michael Addition/Annulation Cascade
Chen, Linlin,Ling, Fei,Liu, Tao,Ma, Yan,Song, Dingguo,Xiao, Lian,Xu, Min,Yu, Mengyao,Zhong, Weihui
, p. 3224 - 3233 (2020/03/23)
We describe here a Cu-catalyzed and 4-OH-TEMPO-mediated sequential dehydrogenation/aza-Michael addition/annulation cascade reaction for the construction of N-alkyl 2-arylindoles from facilely available saturated ketones and 2-arylethynylanilines. This rea
One-pot gold-catalyzed aminofluorination of unprotected 2-alkynylanilines
Arcadi, Antonio,Pietropaolo, Emanuela,Alvino, Antonello,Michelet, Véronique
supporting information, p. 2766 - 2769 (2013/07/19)
A tandem gold(I)-catalyzed aminocylization/fluorination and a two-step, one-pot gold(III)-catalyzed cyclization/electrophilic fluorination provide a convenient and general method for the synthesis of 3,3-difluoro-2-substituted- 3H-indoles in good yield un
