1454771-59-5Relevant articles and documents
Fragment-based discovery of focal adhesion kinase inhibitors
Graedler, Ulrich,Bomke, Joerg,Musil, Djordje,Dresing, Verena,Lehmann, Martin,Hoelzemann, Guenter,Greiner, Hartmut,Esdar, Christina,Krier, Mireille,Heinrich, Timo
, p. 5401 - 5409 (2013/09/23)
Chemically diverse fragment hits of focal adhesion kinase (FAK) were discovered by surface plasmon resonance (SPR) screening of our in-house fragment library. Site specific binding of the primary hits was confirmed in a competition setup using a high-affi