166904-09-2Relevant academic research and scientific papers
GLUCOCORTICOID RECEPTOR AGONIST AND IMMUNOCONJUGATES THEREOF
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Paragraph 001046; 001047, (2018/01/17)
Provided herein are glucocorticoid receptor agonist immunoconjugates, glucocorticoid receptor agonists, and methods of using the same, e.g., to treat autoimmune or inflammatory diseases.
Design of mechanism-based inhibitors of transthyretin amyloidosis: Studies with biphenyl ethers and new structural templates
Gupta, Sarika,Chhibber, Manmohan,Sinha, Sharmistha,Surolia, Avadhesha
, p. 5589 - 5599 (2008/03/17)
Transthyretin (TTR), a tetrameric thyroxine (T4) carrier protein, is associated with a variety of amyloid diseases. In this study, we explore the potential of biphenyl ethers (BPE), which are shown to interact with a high affinity to its T4 binding site t
Novel diphenyl ethers: Design, docking studies, synthesis and inhibition of enoyl ACP reductase of Plasmodium falciparum and Escherichia coli
Chhibber, Manmohan,Kumar, Gyanendra,Parasuraman, Prasanna,Ramya,Surolia, Namita,Surolia, Avadhesha
, p. 8086 - 8098 (2007/10/03)
We designed some novel diphenyl ethers and determined their binding energies for Enoyl-Acyl Carrier Protein Reductase (ENR) of Plasmodium falciparum using Autodock. Out of these, we synthesized the promising compounds and tested them for their inhibitory
Synthesis and insecticidal activity of new substituted phenoxychalcones
Mudaliar, Vivek Ravi,Joshi, Vidya
, p. 456 - 457 (2007/10/02)
Substituted acetophenones (1a-d) on condensation with substituted phenoxyaldehydes (2a-d) in the presence of KOH (50percent) and ethanol give new substituted phenoxychalcones (3a-l).Compounds 3b and 3e have been found to be insecticidally active against housefly (Musca domestica nebulo) adults.
