168909-69-1Relevant academic research and scientific papers
Phosphinic acid analogues of GABA. 1. New potent and selective GABA(B) agonists
Froestl,Mickel,Hall,Von Sprecher,Strub,Baumann,Brugger,Gentsch,Jaekel,Olpe,Rihs,Vassout,Waldmeier,Bittiger
, p. 3297 - 3312 (1995)
The antispastic agent and muscle relaxant baclofen 1 is a potent and selective agonist for bicuculline-insensitive GABA(B) receptors. For many years efforts to obtain superior GABA(B) agonists were unsuccessful. We describe the syntheses and biological pr
