19382-37-7Relevant articles and documents
Electrocatalytic Intermolecular C(sp3)-H/N-H Coupling of Methyl N-Heteroaromatics with Amines and Amino Acids: Access to Imidazo-Fused N-Heterocycles
Qian, Peng,Yan, Zicong,Zhou, Zhenghong,Hu, Kangfei,Wang, Jiawei,Li, Zhibin,Zha, Zhenggen,Wang, Zhiyong
supporting information, p. 6359 - 6363 (2018/10/20)
An efficient NH4I-mediated intermolecular annulation of methyl N-heteroaromatics with amines/amino acids was developed by virtue of anodic oxidation, providing a variety of functionalized imidazo-fused N-heterocycles with good to excellent yields. The practicality of this protocol was demonstrated by the readily available starting materials, broad substrate scope, water tolerance, scalability, and the diverse transformations of the electrolysis product.
Natural α-amino acids applied in the synthesis of imidazo[1,5-a ]N-heterocycles under mild conditions
Wang, Qiang,Zhang, Shuai,Guo, Fengfeng,Zhang, Baiqun,Hu, Ping,Wang, Zhiyong
, p. 11161 - 11166 (2013/02/22)
A facile iodine-mediated decarboxylative cyclization from α-amino acids and N-heterocyclic carbaldehydes was developed. By virtue of this method, a series of imidazo[1,5-a]N-heterocycles can be synthesized efficiently under mild conditions. A tentative re