334792-95-9Relevant articles and documents
Tricyclic pharmacophore-based molecules as novel integrin αvβ3 antagonists. Part IV: Preliminary control of αvβ3 selectivity by meta-oriented substitution
Kubota, Dai,Ishikawa, Minoru,Ishikawa, Midori,Yahata, Naokazu,Murakami, Shoichi,Fujishima, Kazuyuki,Kitakaze, Masafumi,Ajito, Keiichi
, p. 4158 - 4181 (2007/10/03)
To establish the in vivo efficacy of αvβ3/αIIbβ3 dual antagonists possessing a tricyclic pharmacophore, a corresponding αvβ3-selective antagonist was required as a control. We initially too