40899-92-1

Upstream product

• 151721-32-3 N-benzenesulfonyl-o-aminobenzaldehyde 
• 197847-57-7 N-[2-(hydroxymethyl)phenyl]benzenesulfonamide 
• 5344-90-1 2-Aminobenzyl alcohol 
• 98-09-9 benzenesulfonyl chloride 
• 40899-71-6 1-benzenesulfonylindole 
• 120-72-9 indole 
• 3770-50-1 2-carbethoxyindole 
• 541-41-3 chloroformic acid ethyl ester 
• 40900-03-6 1-(benzenesulfonyl)-2-lithioindole 

Downstream Products

• 1265231-79-5 [5-amino-1-(2-methyl-1H-benzimidazol-5-yl)-1H-pyrazol-4-yl]-(1-benzenesulfonyl-1H-indol-2-yl) methanone 
• 1265229-25-1 [5-amino-1-(2-methyl-1H-benzimidazol-5-yl)-1H-pyrazol-4-yl](1H-indol-2-yl)methanone 
• 540740-51-0 1-benzenesulfonyl-1H-indole-2-carboxylic acid hydrazide 
• 40899-93-2 1-(phenylsulfonyl)-1H-indole-2-carboxylic acid 

Relevant academic research and scientific papers

N-(piperidin-4-yl)-1H-indole-2-carboxamide derivatives, preparation method thereof, and pharmaceutical composition for use in preventing or treating Urotensin-Ⅱ receptor activity related diseases containing the same as an active ingredient

The present invention relates to N-(piperidin-4-yl)-1H-indole-2-carboxamide derivatives, a preparation method thereof, and a pharmaceutical composition for preventing or treating urotensin-II receptor activity-related diseases comprising the same as activ

One-pot synthesis of 1-phenylsulfonyl-2-aroylindoles

Interaction of phenylsulfonyl-2-aminobenzaldehyde with 2-bromo-1- phenylethanones in the presence of K2CO3 followed by acid-catalyzed dehydration led to the formation of 1-phenylsulfonyl-2-aroylindoles.Copyright Taylor & Francis Group, LLC.

Heterocycles from ylides. Part X.Synthesis of 3-hydroxy-2,3-dihydroindoles by a domino reaction

A domino reaction between 2-N-phenylsulfonylaminobenzaldehyde (1) and sulfonium ylides (2) leads to 3-hydroxy-2,3-dihydroindoles (3) whose structure was confirmed on the basis of analytical and spectroscopic data.

Novel indolyl aryl sulfones active against HIV-1 carrying NNRTI resistance mutations: Synthesis and SAR studies

The potent anti-HIV-1 activities of L-737,126 (2) and PAS sulfones prompted us to design and test against HIV-1 in acutely infected MT-4 cells a number of novel 1- and 3-benzenesulfonylindoles. Indoles belonging to the 1-benzenesulfonyl series were found

Generation and Reactions of 3-Lithio-1-(phenylsulfonyl)indole

Treatment of 1-(phenylsulfonyl)-3-iodoindole (6) with 2 equiv of tert-butyllithium (-100 deg C THF) generates essentially quantitatively 3-lithio-1-(phenylsulfonyl)indole (1).Quenching 1 with various electrophiles gives 3-substituted indoles in good yield