4196-37-6Relevant academic research and scientific papers
Synthesis of glycosyl-isoindigo derivatives
Sassatelli, Mathieu,Saab, Elias,Anizon, Fabrice,Prudhomme, Michelle,Moreau, Pascale
, p. 4827 - 4830 (2004)
The synthesis of 1-(β-D-glucopyranosyl)-isoindigo from commercially available indoline is described. The synthetic pathway used allowed the substitution of the aromatic moiety by either electron donor or acceptor substituents.
Synthesis and antiproliferative evaluation of glucosylated pyrazole analogs of K252c
Douara, Bachir,Esvan, Yannick J.,Pereira, Elisabeth,Giraud, Francis,Volodina, Yulia L.,Kaluzhny, Dmitry N.,Shtil, Alexander A.,Anizon, Fabrice,Moreau, Pascale
, p. 892 - 901 (2018/01/27)
Pyrazole analogs of the staurosporine aglycon K252c were recently described as potent inhibitors of the three Pim protein kinase isoforms. To evaluate the impact of the introduction of a sugar moiety on the biological activities of this heterocyclic scaffold, four new glucosylated pyrazole analogs of K252c were synthesized. Their biological evaluation demonstrated that most active compounds 11 and 19 substituted by a β-D-glucosyl moiety at N12 or N13 positions exhibited antiproliferative activities toward HCT116 cells.
Synthesis and antiproliferative activities of diversely substituted glycosyl-isoindigo derivatives
Sassatelli, Mathieu,Bouchikhi, Fadoua,Messaoudi, Samir,Anizon, Fabrice,Debiton, Eric,Barthomeuf, Chantal,Prudhomme, Michelle,Moreau, Pascale
, p. 88 - 100 (2007/10/03)
In the course of structure-activity relationship studies, diversely substituted 1-(β-D-glucopyranosyl)-isoindigo derivatives were prepared from commercially available indolines. Their antiproliferative activities were evaluated toward a panel of human solid cancer cell lines (PC 3, DLD-1, MCF-7, M4Beu, A549, PA 1), a murine cell line (L929) and a human fibroblast primary culture to get an insight into the substitution pattern required for the best biological potencies.
Synthesis and biological evaluation of oxindoles and benzimidazolinones derivatives
Messaoudi, Samir,Sancelme, Martine,Polard-Housset, Valerie,Aboab, Bettina,Moreau, Pascale,Prudhomme, Michelle
, p. 453 - 458 (2007/10/03)
The synthesis of new oxindoles and benzimidazolinones derivatives bearing a sugar residue on the aromatic nitrogen is described. The presence of the glycoside moiety should enhance the solubility of these heterocyclic compounds and/or improve the interact
