4912-55-4Relevant academic research and scientific papers
Iron-Catalyzed Intramolecular Aminations of C(sp3)?H Bonds in Alkylaryl Azides
Alt, Isabel T.,Guttroff, Claudia,Plietker, Bernd
supporting information, p. 10582 - 10586 (2017/08/22)
The nucleophilic iron complex Bu4N[Fe(CO)3(NO)] (TBA[Fe]) catalyzes the direct intramolecular amination of unactivated C(sp3)?H bonds in alkylaryl azides, which results in the formation of substituted indoline and tetrahydroquinoline derivatives.
HETEROARYL DERIVATIVES AS SEPIAPTERIN REDUCTASE INHIBITORS
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Paragraph 00146-00150, (2017/05/31)
Inhibitors of sepiapterin reductase of formula (I) or (I'), wherein the substituents are defined as in the claims, and uses of sepiapterin reductase inhibitors in analgesia, treatment of acute and chronic pain, anti-inflammation, and immune cell regulation are disclosed.
NOVEL COMPOUNDS
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Page/Page column 48-49, (2011/02/18)
The present invention relates to new CGRP-antagonists of general formula I wherein U, V, X, Y, R1, R2, R3 and R4 are defined as in the description, the tautomers, the isomers, the diastereomers, the enantiomers, the hydrates, the mixtures thereof and the salts thereof and the hydrates of the salts, particularly the physiologically acceptable salts thereof with inorganic or organic acids or bases, medicaments containing these compounds, their use and processes for preparing them.
DIPOLE STABILIZED α-AMINO-CARBANIONS. III. METALATION-ALKYLATION OF INDOLINES, TETRAHYDROQUINOLINES AND N-METHYLANILINES.
Meyers, A. I.,Hellring, Stuart
, p. 5119 - 5122 (2007/10/02)
Metalation of the 2-position in indolines and tetrahydroquinolines is feasible via their formamidine derivatives using tert-butyllithium.The N-methyl group in N-methylanilines is also metalated using this base.
