52329-04-1Relevant academic research and scientific papers
POLYCYCLIC AMIDES AS UBE2K MODULATORS FOR TREATING CANCER
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Paragraph 00189; 00192-00193, (2021/07/10)
Provided are compounds of Formula (I) and pharmaceutically acceptable salts and compositions thereof, which are useful for treating conditions associated with modulation of UBE2K.
BIARYL-PROPIONIC ACID DERIVATIVES AND THEIR USE AS PHARMACEUTICALS
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Page/Page column 48, (2014/10/15)
The present invention relates to compounds of the formula (I), wherein X, R, R1, R2, D, E1, E2, E3, E4, G1, G2, G3 and G4 have the meanings indicated in the claims, which are valuable pharmaceutical active compounds. They are inhibitors of the protease ca
Biaryl-propionic acid derivatives and their use as pharmaceuticals
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Paragraph 0130; 0131, (2014/10/16)
The present invention relates to compounds of the formula I, wherein X, R, R1, R2, D, E1, E2, E3, E4, G1, G2, G3 and G4 have the meanings indicated in the claims, which are valuable pharmaceutical active compounds. They are inhibitors of the protease cath
BIARYL-PROPIONIC ACID DERIVATIVES AND THEIR USE AS PHARMACEUTICALS
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Page/Page column 48, (2014/10/15)
The present invention relates to compounds of the formula (I), wherein X, R, R1, R2, D, E1, E2, E3, E4, G1, G2, G3 and G4 have the meanings indicated in the claims, which are valuable pharmaceutical active compounds. They are inhibitors of the protease ca
Biaryl-Propionic Acid Derivatives and their Use as Pharmaceuticals
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Paragraph 0140; 0141, (2014/10/16)
The present invention relates to compounds of the formula I, wherein X, R, R1, R2, D, E1, E2, E3, E4, G1, G2, G3 and G4 have the meanings indicated in the claims, which are valuable pharmaceutical active compounds. They are inhibitors of the protease cath
IMIDAZOPYRIDINE COMPOUNDS
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Page/Page column 23, (2010/04/23)
Compounds, pharmaceutical compositions, kits and methods are provided for use with glucokinase that comprise a compound selected from the group consisting of formula (I) wherein the variables are as defined herein.
SYNTHESIS OF PEPTIDE ALKALOIDS-III. AMINO ACIDS AND PEPTIDES-XXXII. SYNTHESIS OF DIHYDRO-ZIZYPHINE A AND B
Schmidt, Ulrich,Boekens, Hilmar,Lieberknecht, Albrecht,Griesser, Helmut
, p. 4949 - 4952 (2007/10/02)
Recently we described a new cyclisation method for the synthesis of ansa peptides by hydrogenolysis of Z-pentafluorophenyl ester and ring closure on the surface of the palladium catalyst.We applied this reaction to the synthesis of the 14-membered ansa pe
