57245-30-4Relevant academic research and scientific papers
New herbicide models from benzoxazinones: Aromatic ring functionalization effects
Macias, Francisco A.,De Siqueira, Joao M.,Chinchilla, Nuria,Marin, David,Varela, Rosa M.,Molinillo, Jose M. G.
, p. 9843 - 9851 (2006)
The utility of benzoxazinones and some of their synthetic derivatives in the search for new leads for herbicide model development has been widely discussed. As the benzoxazinone skeleton contains three different potential areas for functionalization (C-2,
FUSED IMIDAZOLE AND PYRAZOLE DERIVATIVES AS MODULATORS OF TNF ACTIVITY
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Page/Page column 107; 173, (2015/06/25)
A series of substituted benzimidazole, imidazo[1,2-a]pyridine and pyrazolo[1,5-a]pyridine derivatives, and analogues thereof, being potent modulators of human TNFα activity, are accordingly of benefit in the treatment and/or prevention of various human ailments, including autoimmune and inflammatory disorders; neurological and neurodegenerative disorders; pain and nociceptive disorders; cardiovascular disorders; metabolic disorders; ocular disorders; and oncological disorders.
Combined strategy for phytotoxicity enhancement of benzoxazinones
MacIas, Francisco A.,Chinchilla, Nuria,Arroyo, Elena,Molinillo, Jose M. G.,Marin, David,Varela, Rosa M.
experimental part, p. 2047 - 2053 (2010/09/09)
Fifteen new derivatives of D-DIBOA, including aromatic ring modifications and the addition of side chains in positions C-2 and N-4, were synthesized and their phototoxicity, selectivity, and structure-activity relationships evaluated. The most active comp
Synthesis and antimicrobial activity of some new 4-hydroxy-2H-1,4-benzoxazin-3(4H)-ones
Oezden, Seckin,Oeztuerk, Aydin Murat,Goeker, Hakan,Altanlar, Nurten
, p. 715 - 718 (2007/10/03)
Some 4-hydroxy-2H-1,4-benzoxazin-3(4H)-ones were synthesized and evaluated for their antimicrobial activities against Staphylococcus aureus, Escherichia coli and Candida albicans. Compounds 9, and 10 exhibited the best activity against Candida albicans. C
Morpholine derivatives
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, (2008/06/13)
The disclosure relates to new morpholine derivatives which possess antidepressant activity, to processes for the manufacture of said derivatives and to pharmaceutical compositions containing them. Typical of the morpholine derivatives disclosed is 2-(4H-2
