5821-66-9Relevant academic research and scientific papers
An approach to the design of brain-penetrating histaminergic agonists
Young,Ganellin,Griffiths,Mitchell,Parsons,Saunders,Sore
, p. 201 - 211 (1993)
Known and novel histaminergic H1- and H2-receptor agonists were investigated as potentially potent and selective brain-penetrating compounds. Structural modifications were introduced in an attempt to favour passive diffusion across t
Multiple labeling of a potent CX3CR1 antagonist for the treatment of multiple sclerosis
Malmquist, Jonas,Stroem, Peter
, p. 387 - 392,6 (2020/08/24)
Several methods for the preparation of five isotopologues of the CX 3CR1 antagonist 1 were developed. Volatile and radioactive 1-chloro- and 1-bromo-ethyl-benzene was handled in [2′-14C] and [3′, 5′-3H] labeling of 1. d-Le
