70576-29-3Relevant articles and documents
Nickel-Catalyzed Intramolecular Hydroalkenylation of Imines
Feng, Wei-Min,Li, Tian-Yu,Xiao, Li-Jun,Zhou, Qi-Lin
supporting information, p. 7900 - 7904 (2021/10/12)
A ligand-enabled nickel-catalyzed intramolecular hydroalkenylation of imines with unactivated alkenes has been developed. A variety of five- and six-membered cyclic allylic amines were synthesized in high yields. The use of both wide-bite-angle diphosphine ligand and Br?nsted acid is crucial for realizing the reaction. Preliminary investigation of the asymmetric intramolecular hydroalkenylation of imines shows promising potential for the application of the method in the synthesis of enantio-enriched cyclic allylic amines.
Application of Dehydroabietic Acid in Palladium-Catalysed Enyne Cycloisomerisation
Wu, Na,Li, Ruikun,Cui, Feihu,Pan, Yingming
supporting information, p. 2442 - 2447 (2017/07/22)
Dehydroabietic acid (DAA) promotes palladium(0)-catalysed cyclisations of arene-tethered 1,7-enynols and 1,m-enynoates (m=6,7) to give fused carbocyclic dienes. 6,6,6,5-Tetracyclic lactones are accessible by one-pot cycloisomerisation/Diels–Alder reaction
Pyrazolopyrimidine Macrocycles as Inhibitors of Human Immunodeficiency Virus Replication
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Paragraph 0351; 0357, (2015/09/22)
The disclosure generally relates to compounds of formula I, including compositions and methods for treating human immunodeficiency virus (HIV) infection. The disclosure provides novel inhibitors of HIV, pharmaceutical compositions containing such compound