718614-76-7Relevant academic research and scientific papers
Catalytic Synthesis of 3-Thioindoles Using Bunte Salts as Sulfur Sources under Metal-Free Conditions
Qi, Hong,Zhang, Tongxin,Wan, Kefeng,Luo, Meiming
, p. 4262 - 4268 (2016)
An efficient catalytic method for the synthesis of 3-thioindoles has been successfully developed, which uses odorless, stable, readily available crystalline Bunte salts as the sulfenylating agents, iodine as nonmetallic catalyst, and DMSO as both the oxid
1-Benzyl-3-thioaryl-2-carboxyindoles as potent non-peptide endothelin antagonists
Bunker, Amy M.,Edmunds, Jeremy J.,Berryman, Kent A.,Walker, Donnelle M.,Flynn, Michael A.,Welch, Kathy M.,Doherty, Annette M.
, p. 1367 - 1370 (1996)
Endothelin-1 is a potent vasoconstrictor which is thought to be involved in many human disease states. We have developed a series of indole non- peptide endothelin antagonists which display nanomolar receptor affinity. The representative compound from thi
Preparation method of 3-indole thioether
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Paragraph 0015, (2016/10/08)
According to the invention, Bunte salt is employed as a sulfur source to prepare 3-indole thioether. At a certain temperature, elementary iodine or hydroiodic acid and salts thereof is employed as a catalyst, dimethyl sulfoxide is employed as an oxidant,
3-Sulfenylation of indole-2-carboxylates
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Page 8, (2010/02/07)
A highly efficient one-pot procedure for 3-sulfenilation of indole 2-carboxylates is described. Treatment of thiols with N-chlorosuccinimide at -78° C. in CH2Cl2 affords sulfenyl chlorides in situ that readily react with indole 2-carboxylates to give 3-th
