7200-19-3Relevant academic research and scientific papers
Cross-Dehydrogenating Coupling of Aldehydes with Amines/R-OTBS Ethers by Visible-Light Photoredox Catalysis: Synthesis of Amides, Esters, and Ureas
Pandey, Ganesh,Koley, Suvajit,Talukdar, Ranadeep,Sahani, Pramod Kumar
supporting information, p. 5861 - 5865 (2018/09/21)
A straightforward synthesis of amides, ureas, and esters is reported by visible-light cross-dehydrogenating coupling (CDC) of aldehydes (or amine carbaldehydes) and amines/R-OTBS ethers by photoredox catalysis. The reaction is found to be general and high yielding. A plausible mechanistic pathway has been proposed for these transformations and is supported by appropriate controlled experiments.
Optimization of dipeptidic inhibitors of cathepsin L for improved Toxoplasma gondii selectivity and CNS permeability
Zwicker, Jeffery D.,Diaz, Nicolas A.,Guerra, Alfredo J.,Kirchhoff, Paul D.,Wen, Bo,Sun, Duxin,Carruthers, Vern B.,Larsen, Scott D.
supporting information, p. 1972 - 1980 (2018/04/14)
The neurotropic protozoan Toxoplasma gondii is the second leading cause of death due to foodborne illness in the US, and has been designated as one of five neglected parasitic infections by the Center for Disease Control and Prevention. Currently, no trea
5,6-DIHYDROPHENANTHRIDIN-5-YL AS AN ACTIVATABLE PROTECTING GROUP OF CARBOXYLIC ACID - A DIRECT PREPARATION OF AMIDES FROM 5-ACYL-5,6-DIHYDROPHENANTHRIDINE
Narasaka, Koichi,Hirose, Takuji,Uchimaru, Tadafumi,Mukaiyama, Teruaki
, p. 991 - 992 (2007/10/02)
Various amides are directly prepared from the protected carboxylic acids, 5-acyl-5,6-dihydrophenanthridines, by the reaction with primary amines in the presence of ceric pyridinium chloride and cupric oxide.
