760968-79-4

Upstream product

• 760968-78-3 methyl 5-benzyloxy-2-(4-methylbenzenesulfonylamino)benzoate 
• 394-31-0 2-amino-5-hydroxybenzoic acid 
• 1882-72-0 methyl 2-amino-5-hydroxybenzoate 
• 760968-77-2 methyl 5-hydroxy-2-(4-methylbenzenesulfonylamino)benzoate 

Downstream Products

• 791810-64-5 N-[4-benzyloxy-2-(1-(allyloxydiphenylsilyloxy)but-3-enyl)phenyl]-4-methylbenzenesulfonamide 
• 791810-79-2 (Z)-1,5-diacetoxy-5-[5-benzyloxy-2-(4-methylbenzenesulfonylamino)phenyl]-2-pentene 
• 791810-67-8 N-[4-benzyloxy-2-(1,5-dihydroxy-pent-3-enyl)-phenyl]-4-methyl-benzenesulfonamide 
• 791810-63-4 N-[4-benzyloxy-2-(1-hydroxybut-3-enyl)phenyl]-4-methylbenzenesulfonamide 
• 409093-35-2 5-[5-(tert-butyldimethylsiloxy)-2-(4-methylbenzenesulfonylamino)phenyl]-5-hydroxypent-2-enoic acid methyl ester 
• 760968-80-7 N-(4-benzyloxy-2-formylphenyl)-4-methylbenzenesulfonamide 
• 760968-86-3 {3-[6-benzyloxy-1a-hydroxymethyl-3-(toluene-4-sulfonyl)-1a,2,3,7b-tetrahydro-1-oxa-3-aza-cyclopropa[a]naphthalen-2-yl]-propyl}-carbamic acid tert-butyl ester 
• 760968-85-2 {3-[6-benzyloxy-3-hydroxymethyl-1-(toluene-4-sulfonyl)-1,2-dihydro-quinolin-2-yl]-propyl}-carbamic acid tert-butyl ester 
• 760968-88-5 {3-[6-benzyloxy-3-methylene-4-oxo-1-(toluene-4-sulfonyl)-1,2,3,4-tetrahydro-quinolin-2-yl]-propyl}-carbamic acid tert-butyl ester 
• 760968-87-4 {3-[6-benzyloxy-4-hydroxy-3-methylene-1-(toluene-4-sulfonyl)-1,2,3,4-tetrahydro-quinolin-2-yl]-propyl}-carbamic acid tert-butyl ester 
• 760968-82-9 {3-[6-benzyloxy-3-formyl-1-(toluene-4-sulfonyl)-1,2-dihydro-quinolin-2-yl]-propyl}-carbamic acid tert-butyl ester 

Relevant academic research and scientific papers

Synthetic studies on bradykinin antagonist martinellines: Construction of a pyrrolo[3,2-c]quinoline skeleton using silicon-tether RCM reaction and allylic amination

The pyrrolo[3,2-c]quinoline consisting of a core structure of martinellines, the first naturally occurring heterocycle, was prepared through silicon-tether ring-closing metathesis reaction and intramolecular allylic amination as key steps. Graphical Abstr

New synthesis of a pyrroloquinoline skeleton, the martinelline core, using a tandem Michael-aldol strategy

The pyrroloquinoline moiety of Martinelline, a naturally occurring bradykinin receptor antagonist, has been synthesized from 1,2-dihydroquinoline which was prepared by using a tandem Michael-aldol reaction as a key step.