84638-99-3Relevant academic research and scientific papers
Indole derivatives pharmaceutical preparations based thereon, and β-receptor stimulation therewith
-
, (2008/06/13)
Indole derivatives of Formula I STR1 wherein R1 is hydrogen, alkyl of 1-6 carbon atoms, or benzyl R2 is hydrogen, alkyl of up to 4 carbon atoms, free or esterified hydroxyalkyl of up to 4 carbon atoms, or free, amidated or esterified
β2-Agonists containing metabolically labile groups. II. The influence of ester groups in the aryl system
Albrecht,Heindl,Loge
, p. 57 - 60 (2007/10/02)
β2-Agonists which are derived from alkyl 7-hydroxy-indole-2-carboxylates are highly active bronchodilators. The corresponding carboxylic acids, which can be formed metabolically from the esters, have diminished activity. Thus these compounds ar
