857040-81-4Relevant academic research and scientific papers
Novel pseudopeptides incorporating a benzodiazepine-based turn mimetic - Targeting Mycobacterium tuberculosis ribonucleotide reductase
Nurbo, Johanna,Ericsson, Daniel J.,Rosenstr?m, Ulrika,Muthas, Daniel,Jansson, Anna M.,Lindeberg, Gunnar,Unge, Torsten,Karlén, Anders
, p. 1992 - 2000 (2013/05/08)
Peptides mimicking the C-terminus of the small subunit (R2) of Mycobacterium tuberculosis ribonucleotide reductase (RNR) can compete for binding to the large subunit (R1) and thus inhibit RNR activity. Moreover, it has been suggested that the binding of t
New selective AT2 receptor ligands encompassing a γ-turn mimetic replacing the amino acid residues 4-5 of angiotensin II act as agonists
Rosenstr?m, Ulrika,Sk?ld, Christian,Plouffe, Bianca,Beaudry, Hélène,Lindeberg, Gunnar,Botros, Milad,Nyberg, Fred,Wolf, Gunter,Karlén, Anders,Gallo-Payet, Nicole,Hallberg, Anders
, p. 4009 - 4024 (2007/10/03)
New benzodiazepine-based γ-turn mimetics with one or two amino acid side chains were synthesized. The γ-turn mimetics were incorporated into angiotensin II (Ang II) replacing the Val3-Tyr4-Ile 5 or Tyr4-Ile
