85907-56-8Relevant academic research and scientific papers
A new linker for glucuronylated anticancer prodrugs
Rivault, Freddy,Tranoy-Opalinski, Isabelle,Gesson, Jean-Pierre
, p. 675 - 682 (2004)
The synthesis, enzymatic hydrolysis and self decomposition of model glucuronylated prodrugs, incorporating a new linker with different aryl substituents, have been studied. Determination of kinetic parameters (V max, Km and t1/2
NEW STRIGOLACTONE ANALOGS AND THEIR USAGE IN PLANT CONTROL
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Page/Page column 16; 40-41, (2018/04/17)
A strigolactone analog-based composition comprising at least one compound represented by: (I) wherein Ra, Rb, Rc, Rf, Re, and Rz are selected. The compositions can be used in, for example, plant growth regulation and weed control, including controlling th
Synthesis of novel fluorescent 2-{4-[1-(pyridine-2-yl)-1H-pyrazol-3-yl] phenyl}-2H-naphtho [1,2-d] [1,2,3] triazolyl derivatives and evaluation of their thermal and photophysical properties
Padalkar, Vikas S.,Phatangare, Kiran R.,Sekar
, p. 809 - 813 (2013/08/23)
Novel 2-{4-[1-(pyridine-2-yl)-1H-pyrazol-3-yl] phenyl}-2H-naphtho [1,2-d] [1,2,3] triazolyl fluorescent derivatives were synthesized from p-nitrophenylacetic acid and 2-hydrazino pyridine through Vilsmeier-Haack and diazotization reactions. Photophysical properties were evaluated, and results show that compounds have good fluorescence quantum yields. Thermal analysis showed that they are reasonably stable. The structures of the compounds were confirmed by FT-IR, 1H NMR, 13C NMR, and mass spectral and elemental analysis.
β-Heteroarylethyl Groups - New Phosphate-Protecting Groups for Phosphotriester Chemistry
Reiner, Tilman,Kvasyuk, Evgeny,Pfleiderer, Wolfgang
, p. 3053 - 3063 (2007/10/03)
The β-heteroaryl-substituted ethanols 6-10 were synthesized and, together with pyridine-2-ethanols and pyridine-4-ethanols, were tested as a new type of phosphate-protecting groups in the synthesis of oligonucleotides by the phosphotriester approach. The synthesis of 5'-O-(monomethoxytrityl)thymidine 3'-(β-heteroarylethyl 2,5-dichlorophenyl phosphates) 13-17 and 21 provided useful monomeric building blocks in which the various blocking groups could be removed selectively by acid (MeOTr), oximate (2,5-dichlorophenyl phosphate), and 1,8-diazabicyclo[5.4.0]undec-7-ene (DBU) (heteroarylethyl phosphate) treatment. The new, fully blocked dimers 38-41, with β-heteroarylethyl protecting groups in the phosphate moiety, were synthesized. The β-heteroarylethyl groups show a broad range of stability towards base treatment in aprotic solvents depending upon the activation of the H-C(β) atoms by the heterocyclic moiety.
New cardiotonic agents related to amrinone: Synthesis of 1,2-dihydro-5-arylpyridin-2-ones
Gomez-Parra,Del Carmen Gomez,Sanchez,Stefani
, p. 483 - 490 (2007/10/02)
For development of new cardiotonic agents a serie of 5-aryl-3,4-dihydropyridin-2(1H)-ones, related to amrinone have been prepared from methylquinolines, 2-arylacetic acid or 3-arylethanones by direct aminomethylenation and subsequent condensation-cyclizat
Method for inducing tillering utilizing certain pyridine-1-oxides
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, (2008/06/13)
This invention relates to a method of inducing tillering in cereal plants using certain 5-phenyl-3-pyridinecarboxylate compounds, to certain of the compounds themselves, to a process for preparing these compounds, and to agricultural compositions containing them. The compounds are also useful as intermediates for preparing other of the compounds.
Substituted 6-phenyl-1,2,4-triazolo[4,3-a]pyridines
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, (2008/06/13)
This disclosure describes novel 6-(substituted-phenyl)-1,2,4-triazolo[4,3-a]pyridines useful as hypotensive agents.
Substituted 3-alkyl-6-phenyl-1,2,4-triazolo-[4,3-a]pyridines
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, (2008/06/13)
This disclosure describes novel 3-alkyl-6-(substituted-phenyl)-1,2,4-triazolo[4,3-a]pyridines useful as anxiolytic agents.
