956316-86-2

Upstream product

• 459-57-4 4-fluorobenzaldehyde 
• 82891-99-4 ethylene ketal of 3-nitropropanal 
• 956316-85-1 benzyl 3-(2-isopropylhydrazono)propylcarbamate 
• 70629-60-6 isopropylhydrazine hydrochloride 
• 65564-05-8 3-[(benzyloxycarbonyl)amino]propanal 

Downstream Products

• 956316-87-3 3-(4-fluoro-phenyl)-2-isopropyl-7,8-dihydro-2H-1,2,6-triaza-azulene-6-carboxylic acid benzyl ester 
• 851375-22-9 3-(4-fluorophenyl)-2-isopropyl-2,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 
• 1311165-08-8 2-(5-(4-fluorophenyl)-4-(2-(3-(4-fluorophenyl)-2-isopropyl-2,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepin-4-yl)ethyl)-1-isopropyl-1H-pyrazol-3-yl)ethanamine 

Relevant academic research and scientific papers

Convergent synthesis of a 5HT7/5HT2 dual antagonist

The development of an efficient and convergent route to 3-(4-fluorophenyl)-2-isopropyl-2,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine (1), a potent 5HT7/5HT2 dual antagonist, is described. Significant features of this route are: (a) a r

METHODS FOR THE PREPARATION OF PYRAZOLE-CONTAINING COMPOUNDS

The present invention is directed to novel processes for the preparation of fused pyrazole compounds, useful for the treatment of disorders and conditions mediated by serotonin receptor activity.