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Upstream product

• 123-75-1 pyrrolidine 
• 2196-99-8 2-chloro-1-(4-methoxyphenyl)ethanone 
• 6388-72-3 2-(4-methoxyphenyl)oxirane 
• 487012-28-2 1-(4-methoxy-phenyl)-2-pyrrolidin-1-yl-ethanone 
• 120-94-5 1-Methylpyrrolidine 
• 123-11-5 4-methoxy-benzaldehyde 
• 2632-13-5 2-Bromo-4'-methoxyacetophenone 

Relevant academic research and scientific papers

Radical hydroxyalkylation of C-H bond adjacent to nitrogen of tertiary amides, ureas, and amines

Tertiary amides, ureas, and amines undergo direct intermolecular addition to aldehydes under the Et3B/air conditions, thereby providing a unique and simple means for the radical sp3 C-H transformation of nitrogen-containing molecules. Copyright

Synthesis and Biological activity of kappa opioid receptor agonists. Part 2: Preparation of 3-aryl-2-pyridone analogues generated by solution- and solid-phase parallel synthesis methods

New analogues of the previously described 3-aryl pyridone KOR agonists have been synthesised by parallel synthetic methods, both in solution- and with solid-phase chemistry, making use of the well known and versatile Mitsunobu, Suzuki and Buchwald reactions. Opioid receptor binding data for the compounds produced is reported.