98276-57-4

Basic information

• Product Name: 2,4-DIAMINOBENZALDEHYDE
• Synonyms: 2,4-DIAMINOBENZALDEHYDE;Benzaldehyde, 2,4-diamino- (6CI, 9CI);Benzaldehyde, 2,4-diaMino-;4-Formylbenzene-1,3-diamine
• CAS NO: 98276-57-4
• Molecular Formula: C₇H₈N₂O
• Molecular Weight: 136.15
• Product Categories: ALDEHYDE;Aromatic Aldehydes & Derivatives (substituted)
• Mol File: 98276-57-4.mol

Chemical Properties

• Melting Point: 152℃
• Boiling Point: 364.0±32.0 °C(Predicted)
• Appearance: /
• Density: 1.288±0.06 g/cm3(Predicted)
• Storage Temp.: under inert gas (nitrogen or Argon) at 2–8 °C
• PKA: 1.86±0.10(Predicted)
• CAS DataBase Reference: 2,4-DIAMINOBENZALDEHYDE(CAS DataBase Reference)
• NIST Chemistry Reference: 2,4-DIAMINOBENZALDEHYDE(98276-57-4)
• EPA Substance Registry System: 2,4-DIAMINOBENZALDEHYDE(98276-57-4)

Safety Data

• Hazardous Substances Data: 98276-57-4(Hazardous Substances Data)

Usage

Uses

Used in Pharmaceutical Industry:
2,4-DIAMINOBENZALDEHYDE is used as a reagent for the synthesis of various pharmaceutical compounds. One of its applications is in the preparation of 6-(trifluoromethyl)-N-(4-oxothiazolidin-3-yl)quinazoline-2-carboxamide derivatives, which are considered potential DprE1 inhibitors. These inhibitors are significant in the development of new drugs targeting bacterial infections, particularly those caused by drug-resistant strains.

Upstream product

• 528-75-6 2,4-dinitrobenzaldehyde 
• 119-32-4 4-Methyl-3-nitroanilin 
• 100796-40-5 4-acetylamino-1-diacetoxymethyl-2-nitro-benzene 
• 109466-84-4 4-nitro-2-aminobenzaldehyde 
• 102170-39-8 4-amino-2-nitrobenzaldehyde 

Downstream Products

• 1224728-33-9 N-(3-amino-4-formylphenyl)-1-hydroxy-2,2,5,5-tetramethyl-3-pyrrolin-1-oxyl-3-carboxamide 
• 1029773-05-4 7-amino-2-(4-fluorophenyl)quinoline 
• 339538-56-6 4'-trifluoromethyl-biphenyl-2-carboxylic acid (3-amino-4-formyl-phenyl)-amide 
• 67911-35-7 2-Amino-4-(acetylamino)benzaldehyde 
• 109581-97-7 11-amino-20(RS)-camptothecin 

Relevant articles and documents

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